2. Signaling Pathways
  3. GPCR/G Protein
  4. Adenosine Receptor
  5. Adenosine Receptor Isoform
  6. Adenosine Receptor Activator

Adenosine Receptor Activator

Adenosine Receptor Activators (3):

Cat. No. Product Name Effect Purity
  • HY-106199
    Adenosine A1 receptor activator T62
    		Activator 98.93%
    Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor. Adenosine A1 receptor activator T62 produces antinociception in animal models of acute pain and also reduces hypersensitivity in models of inflammatory and nerve-injury pain.
  • HY-161418
    1-NBX
    		Activator
    1-NBX is a potent and selective A1R ligand. 1-NBX exhibits significantly improved A1R affinity with with a Ki of 2.6 nM and lower affinity for the A2A receptor with a Ki of 164 nM. [18F]1-NBX as a promising candidate for further preclinical evaluation as potential PET tracer for A1R imaging.
  • HY-103188
    PD81723
    		Activator
    PD81723 is an adenosine receptor binding enhancer. PD81723 enhances the inhibition of exogenous adenosine in a dose-dependent manner in hippocampal brain sections.